Name and surname:
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Mgr. Peter Šramel, PhD.
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Document type:
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Research/art/teacher profile of a person
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The name of the university:
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Comenius University Bratislava
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The seat of the university:
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Šafárikovo námestie 6, 818 06 Bratislava
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III.a - Occupation-position | III.b - Institution | III.c - Duration |
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Assistant Professor | Comenius University in Bratislava, Faculty of Natural Sciences | 2018 - present (unpaid leave) |
Scientist (part-time) | Centre of experimental medicine, SAS | 2019 - present (unpaid leave) |
Scientist | University of Pardubice, Faculty of chemical technology | 2024 - present |
IV.a - Activity description, course name, other | IV.b - Name of the institution | IV.c - Year |
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Basics in the Python programming language | ITCourse, SAS | 2021 |
Training School, COST Action CM1106 | Universidade de Lisboa, Lisbon, Portugal | 2015 |
X EWDD, European Workshop in Drug Design | Università degli Studi di Siena, Siena, Italy | 2015 |
V.5.a - Name of the course | V.5.b - Study programme | V.5.c - Degree | V.5.d - Field of study |
---|---|---|---|
Bioorganic chemistry (2) | Organic and bioorganic chemistry | 1. Mgr | 17. chemistry |
Krátky, M.; Šramel, P.; Boďo, P.; Šoltésová-Prnová, M.; Kováčiková, L., Májeková, M.; Vinšová, J.; Štefek, M. Novel Rhodanine-based Inhibitors of Aldose Reductase of non-Acidic Nature with P-Hydroxybenzylidene Functional Group. Eur. J. Med. Chem. 2023, 246, 114922, DOI: 10.1016/j.ejmech.2022.114922.
Hlaváč, M.; Kováčiková, L.; Prnová Šoltésová, M.; Šramel, P.; Addová, G.; Májeková, M.; Hanquet, G.; Boháč, A.; Štefek, M. Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur / Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity. J. Med. Chem. 2020, 63, 369 – 381, DOI: 10.1021/acs.jmedchem.9b01747.
Murár, M.; Dobiaš, J.; Šramel, P.; Addová, G.; Hanquet, G.; Boháč, A. Novel CLK1 Inhibitors Based on N-Aryloxazol-2-amine Skeleton – A Possible Way to Dual VEGFR2 TK / CLK Ligands. Eur. J. Med. Chem. 2017, 126, 754 – 761, DOI: 10.1016//j.ejmech.2016.11.003.
Krátky, M.; Šramel, P.; Boďo, P.; Šoltésová-Prnová, M.; Kováčiková, L., Májeková, M.; Vinšová, J.; Štefek, M. Novel Rhodanine-based Inhibitors of Aldose Reductase of non-Acidic Nature with P-Hydroxybenzylidene Functional Group. Eur. J. Med. Chem. 2023, 246, 114922, DOI: 10.1016/j.ejmech.2022.114922.
Hlaváč, M.; Kováčiková, L.; Prnová Šoltésová, M.; Šramel, P.; Addová, G.; Májeková, M.; Hanquet, G.; Boháč, A.; Štefek, M. Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur / Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity. J. Med. Chem. 2020, 63, 369 - 381, DOI: 10.1021/acs.jmedchem.9b01747.
Murár, M.; Dobiaš, J.; Šramel, P.; Addová, G.; Hanquet, G.; Boháč, A. Novel CLK1 Inhibitors Based on N-Aryloxazol-2-amine Skeleton – A Possible Way to Dual VEGFR2 TK / CLK Ligands. Eur. J. Med. Chem. 2017, 126, 754 - 761, DOI: 10.1016//j.ejmech.2016.11.003.
Song, M.; Pang, L.; Zhang, M.; Qu, Y.; Laster Vaughn, K.; Dong, Z. Cdc2-like Kinases: Structure, Biological Function and Therapautic Targets for Diseases. Sig. Transduct. Target. Ther. 2023, 8, 148, DOI: 10.1038/s41392-023-01409-4.
Qin, Z.; Qin, L.; Feng, Xi.; Li, Z.; Bian, J. Developement of Cdc2-like Kinase 2 Inhibitors: Achievments and Future Directions. J. Med. Chem. 2021, 64, 13191 - 13211, DOI: 10.1021/acs.jmedchem.1c00985.
Zhao, W.-H.; Xu, J.-H.; Tangandanchu, V. K. R.; Zhou, C.-H. Thiazolyl Hydrazineylidenyl Indolones as Unique Potential Multitargeting Broad-Spectrum Antimicrobial Agents. Eur. J. Med. Chem. 2023, 256, 115452, DOI: 10.1016/j.ejmech.2023.115452.
Yang, T.; Yang, Y.; Chen, Y.; Tang, M.; Shi, M.; Tian, Y.; Yuan, X.; Yang, Z.; Chen, L. Rational Design and Appraisal of Selective Cdc2-Like Kinase 1 (Clk1) Inhibitors as Novel Autophagy Inducers for the Treatment of Acute Liver Injury (ALI). Eur. J. Med. Chem. 2023, 250, 115168, DOI: 10.1016/j.ejmech.2023.115168.
Kousaxidis, A.; Petrou, A.; Lavrentaki, V.; Fesatidou, M.; Nicolaou, I.; Geronikaki, A. Aldose Reductase and Protein Tyrosine Phosphatase 1B Inhibitors as a Promising Therapeutic Approach for Diabetes Mellitus. Eur. J. Med. Chem. 2020, 207, 112742, DOI: 10.1016/j.ejmech.2020.112742.
Fine organometallic compounds for the green synthesis and catalysis; 2022; APVV-22-0167
A multi-target approach to the diverse molecular mechanisms of diabetic complications and other diseases related to glucose toxicity; 2020; APVV-20-0543
Ligand induced modulation of calcium pump SERCA - study of mechanism and design of new compounds; 2022 - 2026; VEGA 2/0103/22
New substances for the prevention and therapy of diseases caused by glucose toxicity; 2018 - 2021; VEGA 2/0127/18
Medicinal chemistry - an eficient development of inhibitors of selected key biological targets connected with tumor progression; 2018 - 2021; VEGA 1/0670/18
VIII.a - Name of the institution | VIII.b - Address of the institution | VIII.c - Duration (indicate the duration of stay) | VIII.d - Mobility scheme, employment contract, other (describe) |
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Université de Strasbourg, ECPM | 25 Rue Becquerel, 67087, Strasbourg, France | 2014-2017 (total of 21 months) | Co-tutelle de Thése (PhD study under double supervision) |
University of Pardubice, Faculty of chemical technology | Studentská 95, 532 10, Pardubice, Czech republic | 2024 - present | Postdoc |
An author of the Chemistry Olympiad tasks (home, school and regional round), Organic Chemistry, cat, B, 2020 - present
A teaching experience in advanced organic chemistry excercises at a foreign university (Université de Strasbourg, ECPM, France), 2014 - 2016