Name and surname:
|
prof. RNDr. Katarína Mikušová, DrSc.
|
Document type:
|
Research/art/teacher profile of a person
|
The name of the university:
|
Comenius University Bratislava
|
The seat of the university:
|
Šafárikovo námestie 6, 818 06 Bratislava
|
III.a - Occupation-position | III.b - Institution | III.c - Duration |
---|---|---|
head of the department of biochemistry | Comenius University in Bratislava, Faculty of Natural Sciences | 2012 - present |
associate professor | Comenius University in Bratislava, Faculty of Natural Sciences | 2005 - 2022 |
assistent professor | Comenius University in Bratislava, Faculty of Natural Sciences | 1995-2005 |
research assistant | Colorado State University, Fort Collins, USA | 1992-1995 |
university teacher - assistant | Comenius University in Bratislava, Faculty of Natural Sciences | 1988-1989 |
professor | Comenius University in Bratislava, Faculty of Natural Sciences | 2022 - present |
V.1.a - Name of the profile course | V.1.b - Study programme | V.1.c - Degree | V.1.d - Field of study |
---|---|---|---|
Biochemistry (2) | biochemistry | 1. | chemistry |
Biochemistry - Bachelor's thesis (2) | biochemistry | 1 | chemistry |
Biochemistry - Master's thesis (1) | biochemistry | 2 | chemistry |
Laboratory practice | biochemistry | 2 | chemistry |
Biochemistry and molecular biology - selected chapters | biochemistry | 2 | chemistry |
Biochemistry - Master's thesis (1) | biochemistry | 2 | chemistry |
Advanced biochemistry | biochemistry | 3 | chemistry |
Biochemistry (1) | biochemistry | 1. | chemistry |
V.2.a - Name of the study programme | V.2.b - Degree | V.2.c - Field of study |
---|---|---|
Biochemistry | 1 | Chemistry |
Biochemistry (convers.) | 1 | Chemistry |
Biochemistry | 2 | Chemistry |
Biochemistry | 3 | Chemistry |
V.3.a - Name of the field of habilitation procedure and inaugural procedure | V.3.b - Study field to which it is assigned |
---|---|
Organic Chemistry | Chemistry |
V.5.a - Name of the course | V.5.b - Study programme | V.5.c - Degree | V.5.d - Field of study |
---|---|---|---|
Perspectives of biochemistry | biochemistry | 1 | chemistry |
Elective laboratory practice in biochemistry 1 | biochemistry | 2 | chemistry |
Antibiotics | biochemistry | 2 | chemistry |
Elective laboratory practice in biochemistry 2 | biochemistry | 2 | chemistry |
Doctoral seminar 1 | biochemistry | 3 | chemistry |
Doctoral seminar 3 | biochemistry | 3 | chemistry |
Biochemistry | Biological Chemistry | 1 | chemistry |
Structure and function of biomolecules | Biological Chemistry | 1 | Chemistry |
ADC Mikušová, Katarína - Huang, Hairong - Yagi, Tetsuya - Holsters, Marcelle - Vereecke, Danny - D´Haeze, Wim - Scherman, Michael S. - Brennan, Patrick J. - McNeil, Michael R. - Crick, Dean C. : Decaprenylphosphoryl arabinofuranose, the donorof the D-arabinofuranosyl residues of mycobacterial arabinan, is formed via a two-step epimerization of decaprenylphosphoryl ribose. In: Journal of Bacteriology. - Vol. 187, No. 23 (2005), s. 8020-8025, IF (JCR) 2005=4,167, Citations (109)
ADC Beláňová, Martina - Dianišková, Petronela - Brennan, Patrick J. - Completo, Gladys C. - Rose, Natisha L. - Lowary, Todd L. - Mikušová, Katarína: Galactosyl transferases in mycobacterial cell wall synthesis. In: Journal of Bacteriology. - Vol. 190, No. 3 (2008), p. 1141-1145. - IF (JCR) 2008=3,636 Citations (49)
ADC Makarov, Vadim - Manina, Giulia - Mikušová, Katarína - Moellmann, Ute - Ryabova, Olga - Saint-Joanis, Brigitte - Dhar, Neeraj - Pasca, Maria Rosalia - Buroni, Silvia - Lucarelli, Anna Paola - Milano, Anna - De Rossi, Edda - Beláňová,Martina - Bobovska, Adela - Dianišková, Petronela - Korduláková, Jana - Sala, Claudia - Fullam, Elizabeth - Schneider, Patricia - McKinney, John D. - Brodin, Priscille - Christophe, Thierry - Waddell, Simon - Butcher, Philip - Albrethsen, Jakob - Rosenkrands, Ida - Brosch, Roland - Nandi, Vrinda - Bharath, Sowmya - Gaonkar, Sheshagiri - Shandil, Radha K. - Balasubramanian, Venkataraman - Balganesh, Tanjore - Tyagi, Sandeep - Grosset, Jacques - Riccardi, Giovanna - Cole, Stewart T. : Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis. In: Science. - Vol. 324, No. 5928 (2009), s. 801-804, IF (JCR) 2009=29,747, Citations (387)
ADC Trefzer, Claudia - Škovierová, Henrieta - Buroni, Silvia - Bobovská, Adela - Nenci, Simone - Molteni, Elisabetta - Pojer, Florence - Pasca, Maria R. - Makarov, Vadim - Cole, Stewart T. - Riccardi, Giovanna - Mikušová, Katarína - Johnsson, Kai: Benzothiazinones Are Suicide Inhibitors of Mycobacterial Decaprenylphosphoryl-beta-D-ribofuranose 2 '-Oxidase DprE1. In: Journal of the American Chemical Society. - Vol. 134, No. 2 (2012), s. 912-915, IF (JCR) 2012=10,677 Citations (the 110)
ADC Brecik, Miroslav - Centárová, Ivana - Mukherjee, Raju - Kolly, Gaelle S. - Huszár, Stanislav - Bobovská, Adela - Kilacsková, Emöke - Mokošová, Veronika - Svetlíková, Zuzana - Šarkan, Michal - Neres, Joao - Korduláková, Jana - Cole, Stewart T. - Mikušová, Katarína: DprE1 Is a Vulnerable Tuberculosis Drug Target Due to Its Cell Wall Localization. In: ACS Chemical Biology. - Vol. 10, No. 7 (2015), p. 1631-1636. IF (JCR) 2015=5,090 [2014-5,331] Citations (84)
V3 Fan, Dongguang - Wang, Bin - Stelitano, Giovanni - Savková, Karin - Shi, Rui - Huszár, Stanislav - Han, Quanquan - Mikušová, Katarína - Chiarelli, Laurent Roberto - Lu, Yu - Qiao, Chunhua: Structural and Activity Relationships of 6-Sulfonyl-8-Nitrobenzothiazinones as Antitubercular Agents. In: Journal of Medicinal Chemistry. - Vol. 64, No. 19 (2021), pp. 14526-14539. - IF (JCR) 2021=8.039 Citations (6)
Savkova, K., M. Danchenko, V. Fabianova, J. Bellova, M. Bencurova, S. Huszar, J. Kordulakova, B. Sivakova, P. Barath and K. Mikusova (2024). "Compartmentalization of galactan biosynthesis in mycobacteria." J Biol Chem 300(3): 105768.
ADC Makarov, Vadim - Mikušová, Katarína : Development of Macozinone for TB treatment: An Update.
In: Applied sciences. - Vol. 10, No 7 (2020), s. [1-11], art. no. 2269 [online]. IF (JCR) 2019=2,474 Citations (21)
ADC Liu, Lingfeng - Kong, Chengcheng - Fumagalli, Marco - Savková, Karin - Xu, Yiwen - Huszár, Stanislav - Sammartino, José Camilla - Fan, Dongguang - Chiarelli, Laurent R. - Mikušová,Katarína - Sun, Zhaogang - Qiao, Chunhua: Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents. In: European Journal of Medicinal Chemistry. - Vol. 208 (2020), p. [1-11], Art. No. 112773. IF (JCR) 2019=5.573 Citations (9)
ADC Savkova, Karin - Huszar, Stanislav - Barath, Peter - Pakanova, Zuzana - Kozmon, Stanislav - Vancova, Marie - Tesarova, Martina - Blasko, Jaroslav - Kalinak, Michal - Singh, Vinayak - Kordulakova, Jana - Mikusova, Katarina: An ABC transporter Wzm-Wzt catalyzes translocation of lipid-linked galactan across the plasma membrane in mycobacteria. In: Proc Natl Acad Sci U S A Vol. 118 No. 17, e2023663118 (2021) IF (JCR) 2019=9,412 Citations (2)
ADC Beláňová, Martina - Dianišková, Petronela - Brennan, Patrick J. - Completo, Gladys C. - Rose, Natisha L. - Lowary, Todd L. - Mikušová, Katarína: Galactosyl transferases in mycobacterial cell wall synthesis. In: Journal of Bacteriology. - Vol. 190, No. 3 (2008), p. 1141-1145.
[o1] Cuthbertson, L.; Kos, V.; Whitfield, C., ABC transporters involved in export of cell surface glycoconjugates. Microbiology and Molecular Biology Reviews 2010, 74, 341-62.
ADC Mikušová, Katarína - Huang, Hairong - Yagi, Tetsuya - Holsters, Marcelle - Vereecke, Danny - D´Haeze, Wim - Scherman, Michael S. - Brennan, Patrick J. - McNeil, Michael R. - Crick, Dean C. : Decaprenylphosphoryl arabinofuranose, the donorof the D-arabinofuranosyl residues of mycobacterial arabinan, is formed via a two-step epimerization of decaprenylphosphoryl ribose. In: Journal of Bacteriology. - Vol. 187, No. 23 (2005), s. 8020-8025
[o1] Neres, J.; Pojer, F.; Molteni, E.; Chiarelli, L. R.; Dhar, N.; Boy-Rottger, S.; Buroni, S.; Fullam, E.; Degiacomi, G.; Lucarelli, A. P.; Read, R. J.; Zanoni, G.; Edmondson, D. E.; De Rossi, E.; Pasca, M. R.; McKinney, J. D.; Dyson, P. J.; Riccardi, G.; Mattevi, A.; Cole, S. T.; Binda, C., Structural basis for benzothiazinone-mediated killing of Mycobacterium tuberculosis. Science Translational Medicine 2012, 4, 150ra121.
ADC Makarov, Vadim - Manina, Giulia - Mikušová, Katarína - Moellmann, Ute - Ryabova, Olga - Saint-Joanis, Brigitte - Dhar, Neeraj - Pasca, Maria Rosalia - Buroni, Silvia - Lucarelli, Anna Paola - Milano, Anna - De Rossi, Edda - Beláňová,Martina - Bobovska, Adela - Dianišková, Petronela - Korduláková, Jana - Sala, Claudia - Fullam, Elizabeth - Schneider, Patricia - McKinney, John D. - Brodin, Priscille - Christophe, Thierry - Waddell, Simon - Butcher, Philip - Albrethsen, Jakob - Rosenkrands, Ida - Brosch, Roland - Nandi, Vrinda - Bharath, Sowmya - Gaonkar, Sheshagiri - Shandil, Radha K. - Balasubramanian, Venkataraman - Balganesh, Tanjore - Tyagi, Sandeep - Grosset, Jacques - Riccardi, Giovanna - Cole, Stewart T. : Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis. In: Science. - Vol. 324, No. 5928 (2009), s. 801-804,
[o1] Cheng, Y.; Xie, J.; Lee, K. H.; Gaur, R. L.; Song, A.; Dai, T.; Ren, H.; Wu, J.; Sun, Z.; Banaei, N.; Akin, D.; Rao, J., Rapid and specific labeling of single live Mycobacterium tuberculosis with a dual-targeting fluorogenic probe. Science Translational Medicine 2018, 10 (454).
ADC Trefzer, Claudia - Škovierová, Henrieta - Buroni, Silvia - Bobovská, Adela - Nenci, Simone - Molteni, Elisabetta - Pojer, Florence - Pasca, Maria R. - Makarov, Vadim - Cole, Stewart T. - Riccardi, Giovanna - Mikušová, Katarína - Johnsson, Kai: Benzothiazinones Are Suicide Inhibitors of Mycobacterial Decaprenylphosphoryl-beta-D-ribofuranose 2 '-Oxidase DprE1. In: Journal of the American Chemical Society. - Vol. 134, No. 2 (2012), s. 912-915
[o1] Liu, R.; Lyu, X.; Batt, S. M.; Hsu, M. H.; Harbut, M. B.; Vilcheze, C.; Cheng, B.; Ajayi, K.; Yang, B.; Yang, Y.; Guo, H.; Lin, C.; Gan, F.; Wang, C.; Franzblau, S. G.; Jacobs, W. R., Jr.; Besra, G. S.; Johnson, E. F.; Petrassi, M.; Chatterjee, A. K.; Futterer, K.; Wang, F., Determinants of the inhibition of DprE1 and CYP2C9 by antitubercular thiophenes. Angewandte Chemie 2017, 56, 13011-13015.
ADC Brecik, Miroslav - Centárová, Ivana - Mukherjee, Raju - Kolly, Gaelle S. - Huszár, Stanislav - Bobovská, Adela - Kilacsková, Emöke - Mokošová, Veronika - Svetlíková, Zuzana - Šarkan, Michal - Neres, Joao - Korduláková, Jana - Cole, Stewart T. - Mikušová, Katarína: DprE1 Is a Vulnerable Tuberculosis Drug Target Due to Its Cell Wall Localization. In: ACS Chemical Biology. - Vol. 10, No. 7 (2015), p. 1631-1636.
[o1] Bahuguna, A. and D. S. Rawat, An overview of new antitubercular drugs, drug candidates, and their targets. Medicinal Research Reviews 2020, 40, 263-292.
Computer-aided design of novel antituberculosis compounds and their experimental evaluation
APVV 20-0230 (2021-2025)
Investigator (Principal Investigator for the partner institution)
Design, Synthesis and Mode of Action Study of New Original Heterocyclic Compounds with Activity on Latent Tuberculosis Infection;
Ministry of Education, School, Science, Research and Sport of the Slovak Republic, scientific and technical services within the Slovak-Russian cooperation, contract number 0395/2016 (2016 - 2018)
Principal Investigator
Topological aspects of mycobacterial arabinogalactan biosynthesis - functional characterization of selected mycobacterial ABC transporters.
APVV-15-0515 (2016-2020)
Principal Investigator
Investigation of the mechanism of action of antimycobacterial inhibitors - development of a new methodology for the investigation of mechanisms of action of new antimycobacterial compounds;
VEGA 1/0301/18 (2018 – 2021)
Deputy of the principal investigator
Deciphering the final stages of mycobacterial cell wall core biosythesis
Recovery and resilience facility
Project number: 09I01-03-V03-00001 (September 2023 - June 2026
Acronym: MyTB-Core
Principal investigator
VII.a - Activity, position | VII.b - Name of the institution, board | VII.c - Duration |
---|---|---|
Co-guarantee of the Board for the Doctoral Study Program "Biochemistry" | Comenius University in Bratislava, Faculty of Natural Sciences | 2009 - present |
Alternating chairman (previously member) of the state exam committee for Biochemistry master's degree | Comenius University in Bratislava, Faculty of Natural Sciences | 2005 - present |
Member of the state exam committee for Biochemistry bachelor's degree | Comenius University in Bratislava, Faculty of Natural Science | 2005 - present |
Member of the VEGA Evaluation Committee for Chemical Sciences | Ministry of Education, School, Science, Research and Sport of the Slovak Republic | since 2021 |
Chair of the "ad hoc" committee for the defense of doctoral theses in the field of Biochemistry | Ministry of Education, School, Science, Research and Sport of the Slovak Republic | since 2021 |
VIII.a - Name of the institution | VIII.b - Address of the institution | VIII.c - Duration (indicate the duration of stay) | VIII.d - Mobility scheme, employment contract, other (describe) |
---|---|---|---|
Department of Microbiology, Immunology, and Pathology, Colorado State University | Fort Collins, USA | 06/1992-07/1995 | research assistant (work contract) |
Department of Microbiology, Immunology, and Pathology, Colorado State University | Fort Collins, USA | 10 short term stays (1-2 months) between 1996-2008 | visiting scientist - invitation by prof. P.J. Brennan to perform investigation of metabolic pathways of mycobacterial cell wall synthesis |
AstraZeneca | Bangalore, India | 25/09/2006-06/10/2006 | visiting scientist - invitation by Dr. T. Balganesh to perform optimization of high throughput screening of mannosyltransferase PimA |
Member of the Learned Society of Slovakia since 2021