Name and surname:
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Mgr. Stanislav Huszár, PhD.
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Document type:
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Research/art/teacher profile of a person
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The name of the university:
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Comenius University Bratislava
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The seat of the university:
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Šafárikovo námestie 6, 818 06 Bratislava
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III.a - Occupation-position | III.b - Institution | III.c - Duration |
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Assistant professor | Department of Biochemistry, Faculty of Natural Sciences, Comenius University in Bratislava | 2016 - present |
V.1.a - Name of the profile course | V.1.b - Study programme | V.1.c - Degree | V.1.d - Field of study |
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Bachelor Thesis in Biochemistry (2) | Biochemistry | I. | Chemistry |
Biochemistry and Cell Biology Advanced Laboratory Practices | Biochemistry | II. | Chemistry |
Methods in Biochemistry | Biochemistry | I. | Chemistry |
V.5.a - Name of the course | V.5.b - Study programme | V.5.c - Degree | V.5.d - Field of study |
---|---|---|---|
Optional laboratory practice in biochemistry and molecular biology | Biochemistry | II. | Chemistry |
Biochemistry and Cell Biology Laboratory Practices | Biochemistry | I. | Chemistry |
Perspectives in Biochemistry | Biochemistry, Biology | I. | Chemistry |
Bachelor Thesis in Biochemistry (1) | Biochemistry | I. | Chemistry |
Savková, K., Huszár, S., Baráth, P., Pakanová, Z., Kozmon, S., Vancová, M., Tesařová, M., Blaško, J., Kaliňák, M., Singh, V., Korduláková, J., and Mikušová, K. (2021) An ABC transporter Wzm–Wzt catalyzes translocation of lipid-linked galactan across the plasma membrane in mycobacteria. Proc. Natl. Acad. Sci. 118, e2023663118, IF (JCR) 2019=9.412
Citations (4)
Huszár, S., Singh, V., Polčicová, A., Baráth, P., Belén Barrio, M., Lagrange, S., Leblanc, V., Nacy, C. A., Mizrahi, V., and Mikušová, K. (2017) N-Acetylglucosamine-1-Phosphate Transferase, WecA, as a Validated Drug Target in Mycobacterium tuberculosis. Antimicrob. Agents Chemother. 61, 1–16, IF (JCR) 2017=4.255
Citations (19)
Brecik, M., Centárová, I., Mukherjee, R., Kolly, G. S., Huszár, S., Bobovská, A., Kilacsková, E., Mokošová, V., Svetlíková, Z., Šarkan, M., Neres, J., Korduláková, J., Cole, S. T., and Mikušová, K. (2015) DprE1 Is a Vulnerable Tuberculosis Drug Target Due to Its Cell Wall Localization. ACS Chem. Biol. 10, 1631–1636, IF (JCR) 2015=5.090
Citations (126)
Makarov, V., Neres, J., Hartkoorn, R. C., Ryabova, O. B., Kazakova, E., Šarkan, M., Huszár, S., Piton, J., Kolly, G. S., Vocat, A., Conroy, T. M., Mikušová, K., and Cole, S. T. (2015) The 8-Pyrrole-Benzothiazinones Are Noncovalent Inhibitors of DprE1 from Mycobacterium tuberculosis. Antimicrob. Agents Chemother. 59, 4446–4452, IF (JCR) 2015=4.415
Citations (68)
Wang, F., Sambandan, D., Halder, R., Wang, J., Batt, S. M., Weinrick, B., Ahmad, I., Yang, P., Zhang, Y., Kim, J., Hassani, M., Huszar, S., Trefzer, C., Ma, Z., Kaneko, T., Mdluli, K. E., Franzblau, S., Chatterjee, A. K., Johnsson, K., Mikusova, K., Besra, G. S., Futterer, K., Robbins, S. H., Barnes, S. W., Walker, J. R., Jacobs, W. R., and Schultz, P. G. (2013) Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. Proc. Natl. Acad. Sci. 110, E2510–E2517, IF (JCR) 2013=9.809
Citations (188)
Savková, K., Huszár, S., Baráth, P., Pakanová, Z., Kozmon, S., Vancová, M., Tesařová, M., Blaško, J., Kaliňák, M., Singh, V., Korduláková, J., and Mikušová, K. (2021) An ABC transporter Wzm–Wzt catalyzes translocation of lipid-linked galactan across the plasma membrane in mycobacteria. Proc. Natl. Acad. Sci. 118, e2023663118, IF (JCR) 2019=9.412
Citations (4)
Huszár, S., Chibale, K., and Singh, V. (2020) The quest for the holy grail: new antitubercular chemical entities, targets and strategies. Drug Discov. Today. 00, 1–9, IF (JCR) 2019=7.321
Citations (42)
Karabanovich, G., Dušek, J., Savková, K., Pavliš, O., Pávková, I., Korábečný, J., Kučera, T., Kočová Vlčková, H., Huszár, S., Konyariková, Z., Konečná, K., Jand’ourek, O., Stolaříková, J., Korduláková, J., Vávrová, K., Pávek, P., Klimešová, V., Hrabálek, A., Mikušová, K., and Roh, J. (2019) Development of 3,5-Dinitrophenyl-Containing 1,2,4-Triazoles and Their Trifluoromethyl Analogues as Highly Efficient Antitubercular Agents Inhibiting Decaprenylphosphoryl-β- d -ribofuranose 2′-Oxidase . J. Med. Chem. 62, 8115–8139, IF (JRC) 2019=6.205
Citations (38)
Chiarelli, L. R., Mori, G., Orena, B. S., Esposito, M., Lane, T., de Jesus Lopes Ribeiro, A. L., Degiacomi, G., Zemanová, J., Szádocka, S., Huszár, S., Palčeková, Z., Manfredi, M., Gosetti, F., Lelièvre, J., Ballell, L., Kazakova, E., Makarov, V., Marengo, E., Mikusova, K., Cole, S. T., Riccardi, G., Ekins, S., and Pasca, M. R. (2018) A multitarget approach to drug discovery inhibiting Mycobacterium tuberculosis PyrG and PanK. Sci. Rep. 8, 3187, IF (JRC) 2018=4.011
Citations (35)
Huszár, S., Singh, V., Polčicová, A., Baráth, P., Belén Barrio, M., Lagrange, S., Leblanc, V., Nacy, C. A., Mizrahi, V., and Mikušová, K. (2017) N-Acetylglucosamine-1-Phosphate Transferase, WecA, as a Validated Drug Target in Mycobacterium tuberculosis. Antimicrob. Agents Chemother. 61, 1–16, IF (JCR) 2017=4.255
Citations (19)
Wang, F., Sambandan, D., Halder, R., Wang, J., Batt, S. M., Weinrick, B., Ahmad, I., Yang, P., Zhang, Y., Kim, J., Hassani, M., Huszar, S., Trefzer, C., Ma, Z., Kaneko, T., Mdluli, K. E., Franzblau, S., Chatterjee, A. K., Johnsson, K., Mikusova, K., Besra, G. S., Futterer, K., Robbins, S. H., Barnes, S. W., Walker, J. R., Jacobs, W. R., and Schultz, P. G. (2013) Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. Proc. Natl. Acad. Sci. 110, E2510–E2517;
Cit.: Trivedi, A., Mavi, P. S., Bhatt, D., and Kumar, A. (2016) Thiol reductive stress induces cellulose-anchored biofilm formation in Mycobacterium tuberculosis. Nat. Commun. 7, 11392
Wang, F., Sambandan, D., Halder, R., Wang, J., Batt, S. M., Weinrick, B., Ahmad, I., Yang, P., Zhang, Y., Kim, J., Hassani, M., Huszar, S., Trefzer, C., Ma, Z., Kaneko, T., Mdluli, K. E., Franzblau, S., Chatterjee, A. K., Johnsson, K., Mikusova, K., Besra, G. S., Futterer, K., Robbins, S. H., Barnes, S. W., Walker, J. R., Jacobs, W. R., and Schultz, P. G. (2013) Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. Proc. Natl. Acad. Sci. 110, E2510–E2517;
Cit.: Kavvas, E. S., Catoiu, E., Mih, N., Yurkovich, J. T., Seif, Y., Dillon, N., Heckmann, D., Anand, A., Yang, L., Nizet, V., Monk, J. M., and Palsson, B. O. (2018) Machine learning and structural analysis of Mycobacterium tuberculosis pan-genome identifies genetic signatures of antibiotic resistance. Nat. Commun. 9, 4306
Brecik, M., Centárová, I., Mukherjee, R., Kolly, G. S., Huszár, S., Bobovská, A., Kilacsková, E., Mokošová, V., Svetlíková, Z., Šarkan, M., Neres, J., Korduláková, J., Cole, S. T., and Mikušová, K. (2015) DprE1 Is a Vulnerable Tuberculosis Drug Target Due to Its Cell Wall Localization. ACS Chem. Biol. 10, 1631–1636;
Cit.: Warrier, T., Kapilashrami, K., Argyrou, A., Ioerger, T. R., Little, D., Murphye, K. C., Nandakumar, M., Park, S., Gold, B., Mi, J., Zhang, T., Meiler, E., Rees, M., Somersan-Karakaya, S., Francisco, E. P. De, Martinez-Hoyos, M., Burns-Huang, K., Roberts, J., Ling, Y., Rhee, K. Y., Mendoza-Losana, A., Luo, M., and Nathan, C. F. (2016) N-methylation of a bactericidal compound as a resistance mechanism in Mycobacterium tuberculosis. Proc. Natl. Acad. Sci. U. S. A. 113, E4523–E4530
Wang, F., Sambandan, D., Halder, R., Wang, J., Batt, S. M., Weinrick, B., Ahmad, I., Yang, P., Zhang, Y., Kim, J., Hassani, M., Huszar, S., Trefzer, C., Ma, Z., Kaneko, T., Mdluli, K. E., Franzblau, S., Chatterjee, A. K., Johnsson, K., Mikusova, K., Besra, G. S., Futterer, K., Robbins, S. H., Barnes, S. W., Walker, J. R., Jacobs, W. R., and Schultz, P. G. (2013) Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. Proc. Natl. Acad. Sci. 110, E2510–E2517;
Cit.: Richter, A., Rudolph, I., Möllmann, U., Voigt, K., Chung, C., Singh, O. M. P., Rees, M., Mendoza-Losana, A., Bates, R., Ballell, L., Batt, S., Veerapen, N., Fütterer, K., Besra, G., Imming, P., and Argyrou, A. (2018) Novel insight into the reaction of nitro, nitroso and hydroxylamino benzothiazinones and of benzoxacinones with Mycobacterium tuberculosis DprE1. Sci. Rep. 8, 13473
Brecik, M., Centárová, I., Mukherjee, R., Kolly, G. S., Huszár, S., Bobovská, A., Kilacsková, E., Mokošová, V., Svetlíková, Z., Šarkan, M., Neres, J., Korduláková, J., Cole, S. T., and Mikušová, K. (2015) DprE1 Is a Vulnerable Tuberculosis Drug Target Due to Its Cell Wall Localization. ACS Chem. Biol. 10, 1631–1636;
Cit.: Richter, A., Rudolph, I., Möllmann, U., Voigt, K., Chung, C., Singh, O. M. P., Rees, M., Mendoza-Losana, A., Bates, R., Ballell, L., Batt, S., Veerapen, N., Fütterer, K., Besra, G., Imming, P., and Argyrou, A. (2018) Novel insight into the reaction of nitro, nitroso and hydroxylamino benzothiazinones and of benzoxacinones with Mycobacterium tuberculosis DprE1. Sci. Rep. 8, 13473
Grant APVV-19-0189 (2020 - 2024): Activation of drugs against tuberculosis - solving 3D structures of selected activating enzymes and characterization of mechanisms of activation/metabolism of ethionamide, rifampicin and pretomanide; co-investigator
Grant VEGA 1/0781/19 (2019 - 2022): The study of the electron transport chain in Mycobacterium tuberculosis and Diplonema papillatum - development and optimization of new methodologies for monitoring of Mycobacterium tuberculosis and a Diplonema papillatum electron transport chain complexes. Purification and biochemical characterization of mycobacterial cytochrome bd oxidase; principal investigator
Grant VEGA 1/0301/18 (2018 - 2021): Investigation of the mechanism of action of antimycobacterial inhibitors - development of a new methodology for the investigation of mechanisms of action of new antimycobacterial compounds; co-investigator
Grant APVV-15-0515 (2016 - 2020): Topological aspects of mycobacterial arabinogalactan biosynthesis - functional characterization of selected mycobacterial ABC transporters; co-investigator
Grant VEGA 1/0441/15 (2015 - 2017): Biochemical characterization of mycobacterial proteins WecA and MraY - potential targets for antituberculosis drugs; co-investigator
VIII.a - Name of the institution | VIII.b - Address of the institution | VIII.c - Duration (indicate the duration of stay) | VIII.d - Mobility scheme, employment contract, other (describe) |
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Drug Discovery and Development Centre (H3D), University of Cape Town | Rondebosch 7701, Cape Town, Western Cape, South Africa | October - December 2018 | Intership - construction of mycobacterial knockdown strians by CRISPR-Cas |
Drug Discovery and Development Centre (H3D), University of Cape Town | Rondebosch 7701, Cape Town, Western Cape, South Africa | June 2019 - March 2020 | Postdoctoral fellowship |